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Ketamine Pharmacology: An Update – PubMed Central (PMC)

 March 25, 2026

For more than 50 years, ketamine has proven to be a safe anesthetic drug with potent analgesic properties. The active enantiomer is S (+)‐ketamine. Ketamine is mostly metabolized in norketamine, an active metabolite.

https://pmc.ncbi.nlm.nih.gov/articles/PMC6493357/

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